Dec 11 2013
Dostinex (Cabergoline) is one of the most popular drugs to reduce prolactin-related side effects in athletes using anabolic androgenic steroids or other performance enhancing drugs. This dopamine agonist is commonly used in the management of hyperprolactinemia and its symptoms and is equally effective for both men and women.
Dostinex possesses significant affinity for the D3, D4, 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, α2B– receptors, and moderate/low affinity for the D1 and 5-HT7 receptors. This drug functions as an agonist at all receptors except for 5-HT7 and α2B-, where it acts as an antagonist. The tablets of Dostinex include Cabergoline, a dopamine receptor agonist and chemical name of the drug is 1-[(6-allylergolin-8ß-yl)-carbonyl]-1-[3-(dimethylamino) propyl]-3-ethylurea. Its molecular formula is C26H37N5O2, and its molecular weight is 451.62. For oral administration, Dostinex tablets include 0.5 mg of Cabergoline and the list of inactive ingredients includes leucine, USP, lactose, and NF.
Dostinex is also one of the very few drugs that can enhance motor skills quickly and help athletes learn new techniques, methods, or strategies at a faster rate than their competitors. This synthetic ergoline with a high affinity to dopamine D2 receptors demonstrates a strong prolonged activity inhibitor of prolactin secretion.
This drug is commonly used to treat disorders associated with high levels of the hormone prolactin, either due to tumors in the pituitary gland or to unknown causes. It is also prescribed for the treatment of health complications like monotherapy of Parkinson’s disease in the early phase, treatment of uterine fibroids, lower ACTH levels and cause regression of ACTH producing pituitary adenomas, and controlling or reducing other kinds of pituitary adenomas, as well as silent or non-functional adenomas. It may also be prescribed for providing relief to men diagnosed with enlarged mammary glands, production of milk, reduced sperm production, impotency, and decreased sex drive.
One of the biggest advantages of Dostinex is that it allows athletes and bodybuilders to use Deca Durabolin, Anavar and Trenbolone together in a steroid cycle, without any concerns. Since these two steroids are great additions to any cycle, Dostinex proves its worth in an amazing way. In addition to these advantages, Dostinex also has the potential of reducing the time one needs to recover and gain an erection between orgasms by reducing or eliminating the male refractory period. This of course significantly enhances all parameters of sexual function, drive, and satisfaction. Furthermore, this drug is also useful to combat galactorrhea, gynecomastia, and sexual dysfunction. It is also used as a post cycle therapy and recovery drug for combating estrogenic side effects such as oily skin, acne, gynecomastia, and bloating. This drug also has the ability to make athletes feel “full” more often and reduce cravings for food, without feeling the discomfort that dieting usually brings. It is also admired for its potential to help athletes avoid anxiety and discomfort associated with calorie restrictions. Since this drug is not physically and mentally addictive and one of the best drugs to promote the sense of well being, it has been an instant hit with athletes across the world for the last many decades.
The recommended dose of Dostinex for adults is 0.5 mg per week, given in 1 or 2 doses per week. The dose may be increased by 0.5 mg per week until a maximum dose of 2 mg per week is reached. It is very important to note that doses of this drug should not be increased more often than every 4 weeks.
|1||20 mg every day||75 mg every day|
|2||20 mg every day||75 mg every day|
|3||20 mg every day||75 mg every day|
|4||20 mg every day||75 mg every day|
|5||20 mg every day||75 mg every day|
|6||20 mg every day||75 mg every day||50 mg every day|
|7||20 mg every day||75 mg every day||50 mg every day||50 mg every day||1 mg every day|
|8||75 mg every day||50 mg every day||50 mg every day||1 mg every day|
|9||75 mg every day||50 mg every day||50 mg every day||1 mg every day|
|10||75 mg every day||50 mg every day||50 mg every day||1 mg every day|
|11||50 mg every day||50 mg every day||1 mg every day|
Dostinex abuse may lead to health concerns like irregular heartbeat, breathing problems, or leg cramps or pain in the toes or fingers. Medical advice should be sought on an immediate basis after stopping use of this drug in case side effects like weakness, tiredness, breast pain, hot flushes, dizziness, unusual sleepiness, and abdominal pain are experienced after using Dostinex tablets or injections.